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BDBM50005685 2,2-Diphenyl-propionic acid 2-diethylamino-ethyl ester::2,2-Diphenyl-propionic acid 2-diethylamino-ethyl ester(Aprophen)::2-(diethylamino)ethyl 2,2-diphenylpropanoate::Aprofene::Aprophen::CHEMBL26505

SMILES: CCN(CC)CCOC(=O)C(C)(c1ccccc1)c1ccccc1

InChI Key: InChIKey=DIDYGLSKVUKRRP-UHFFFAOYSA-N

Data: 17 KI  2 IC50

Find this compound or compounds like it in BindingDB or PDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 19 hits for monomerid = 50005685   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Pancreatic alpha-amylase


(Rat)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
n/an/a 46n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Carboxylic ester hydrolase


(Horse)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
n/an/a 6.70E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor M1


(Rat)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
0.850n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor M2


(Rat)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
1.70n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor M1


(Human)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
2.10n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor M3


(Rat)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
3.39n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor


(Rabbit)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
3.80n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor M2


(Rat)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
4.90n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor M4


(Chicken)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
5.5n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor M4


(Human)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
7.40n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor M3


(Human)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
7.70n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor M2


(Human)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
9.30n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor M1


(Human)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
15.1n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor M1/M2/M3/M4/M5


(Human)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
23n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor M1


(Human)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
26.5n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic receptor M1


(Bovine)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
51n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor M2


(Human)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
107n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor M4


(Human)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
628n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor M3


(Human)
BDBM50005685
PNG
(Aprophen | 2-(diethylamino)ethyl 2,2-diphenylpropa...)
GoogleScholar
UniChem
7.76E+3n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair