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BDBM35938 1-(p-chlorophenyl)-1-(2-pyridyl)-3-N,N-dimethylpropylamine::1-(p-chlorophenyl)-1-(2-pyridyl)-3-dimethylaminopropane::3-(p-chlorophenyl)-3-(2-pyridyl)-N,N-dimethylpropylamine::5-HT,N-ACETYL::CHEMBL505::CHLORPHENIRAMINE::CHLORPHENIRAMINE MALEATE::Polaramin::Polaramine::Polaronil::[3H]Chlorphenamine::[3H]Chlorpheniramine::chlorophenylpyridamine::chlorphenamine::clorfeniramina::d-Chlorpheniramine::gamma-(4-chlorophenyl)-N,N-dimethyl-2-pyridinepropanamine::gamma-(4-chlorophenyl)-gamma-(2-pyridyl)propyldimethylamine

SMILES: CN(C)CCC(c1ccc(Cl)cc1)c1ccccn1

InChI Key: InChIKey=SOYKEARSMXGVTM-UHFFFAOYSA-N

Data: 25 KI  23 IC50

Find this compound or compounds like it in BindingDB or PDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 48 hits for monomerid = 35938   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Bile salt export pump


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a>1.35E+5n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Lethal(3)malignant brain tumor-like protein 3


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a 4.20E+4n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a 66n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a 1.10E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Guinea pig)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a 12n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a 2.09E+4n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Isoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a 4.10E+4n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
MBT domain-containing protein 1


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a 3.40E+4n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Guinea pig)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a 291n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Guinea pig)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a 8.80n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Lethal(3)malignant brain tumor-like protein 4


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a>1.00E+5n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Platelet-activating factor receptor


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a>5.00E+4n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
ATP-binding cassette sub-family C member 3


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a>1.33E+5n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
ATP-binding cassette sub-family C member 2


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a>1.33E+5n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
ATP-binding cassette sub-family C member 4


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a>1.33E+5n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Bile salt export pump


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a>1.33E+5n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Sodium channel protein type 1/2/3 subunit alpha


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a 1.00E+4n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a 2.09E+4n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a 2.09E+4n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a 2.09E+4n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Solute carrier family 22 member 2


(Rat)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a 2.60E+4n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Solute carrier family 22 member 1


(Rat)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a 1.40E+4n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Chloroquine resistance transporter


(malaria parasite P. falciparum)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
n/an/a 5.40E+4n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Guinea pig)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
0.440n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Guinea pig)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
0.5n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Guinea pig)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
0.690n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Guinea pig)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
1.98n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Rat)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
2n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
2.51n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
2.51n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
2.67n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
4.47n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
4.5n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
4.81n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Rat)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
5.5n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Rat)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
5.5n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
7n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Rat)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
8n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
15n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
30n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H4 receptor


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
2.91E+3n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
5-hydroxytryptamine receptor 2C


(Rat)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
3.12E+3n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
5-hydroxytryptamine receptor 2B


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
4.17E+3n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
5-hydroxytryptamine receptor 2B


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
6.80E+3n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
5-hydroxytryptamine receptor 2B


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
7.22E+3n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
5-hydroxytryptamine receptor 2C


(Human)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
>1.00E+4n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor M2


(Rat)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
>1.00E+4n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Hrh3 protein


(Rat)
BDBM35938
PNG
(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
GoogleScholar
UniChem
>1.00E+4n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair