BDBM50010504 CHEMBL3264371

SMILES Fc1cc(F)cc(c1)N1CCN(CCNC(=O)c2cnc3ccccc3n2)CC1

InChI Key InChIKey=ACOGYNPKOWYKEV-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50010504   

Target5-hydroxytryptamine receptor 1A(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50010504(CHEMBL3264371)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-8-OH-OPAT from human recombinant 5HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50010504(CHEMBL3264371)
Affinity DataIC50: 1.14E+3nMAssay Description:Agonist activity at Wistar rat brain 5HT1A receptor assessed as inhibition of firing rate of dorsal raphe nucleus by electrophysiological analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed