BDBM50011518 CHEMBL3262548

SMILES CCC1C(=O)N(C2CCN(Cc3cccc4[nH]ccc34)CC2)c2ccccc12

InChI Key InChIKey=IHHKRBWQSBPVHH-UHFFFAOYSA-N

Data  3 KI  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50011518   

TargetNociceptin receptor(Homo sapiens (Human))
Astraea Therapeutics

Curated by ChEMBL
LigandPNGBDBM50011518(CHEMBL3262548)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]N/OFQ from human nociceptin opioid receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astraea Therapeutics

Curated by ChEMBL
LigandPNGBDBM50011518(CHEMBL3262548)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor transfected in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astraea Therapeutics

Curated by ChEMBL
LigandPNGBDBM50011518(CHEMBL3262548)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor transfected in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Astraea Therapeutics

Curated by ChEMBL
LigandPNGBDBM50011518(CHEMBL3262548)
Affinity DataEC50:  82nMAssay Description:Agonist activity at human nociceptin opioid receptor transfected in CHO cell membranes assessed as stimulation of [35S]GTPgammaS binding after 60 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Astraea Therapeutics

Curated by ChEMBL
LigandPNGBDBM50011518(CHEMBL3262548)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human mu opioid receptor transfected in CHO cell membranes assessed as stimulation of [35S]GTPgammaS binding after 60 mins by sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astraea Therapeutics

Curated by ChEMBL
LigandPNGBDBM50011518(CHEMBL3262548)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human kappa opioid receptor transfected in CHO cell membranes assessed as stimulation of [35S]GTPgammaS binding after 60 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed