BDBM50011620 2-{3-[1-Ethyl-6-(2-fluoro-phenyl)-4H-2,3,5,10b-tetraaza-benzo[e]azulen-8-yl]-prop-2-ynyl}-isoindole-1,3-dione::CHEMBL283152

SMILES CCc1nnc2CN=C(c3ccccc3F)c3cc(ccc3-n12)C#CCN1C(=O)c2ccccc2C1=O

InChI Key InChIKey=CTRLDMFOIYQMMB-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50011620   

TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011620(2-{3-[1-Ethyl-6-(2-fluoro-phenyl)-4H-2,3,5,10b-tet...)
Affinity DataIC50:  100nMAssay Description:PAF-antagonist activity determined in dog platelets by PAF-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed