BDBM50011647 2-{3-[6-(2-Fluoro-phenyl)-1-methyl-4H,6H-5-oxa-2,3,10b-triaza-benzo[e]azulen-8-yl]-prop-2-ynyl}-isoindole-1,3-dione::CHEMBL282666

SMILES Cc1nnc2COC(c3ccccc3F)c3cc(ccc3-n12)C#CCN1C(=O)c2ccccc2C1=O

InChI Key InChIKey=DBDRVZPLYRUKRB-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50011647   

TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011647(CHEMBL282666 | 2-{3-[6-(2-Fluoro-phenyl)-1-methyl-...)
Affinity DataIC50: 500nMAssay Description:PAF-antagonist activity determined in dog platelets by PAF-binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed