BDBM50019481 CHEMBL2028997::NH2-Tyr-Gly-Gly-Phe-D-Trp-Arg-Arg-D-Trp-Arg-D-Pro-Lys-OH
SMILES CC[C@H](C)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(O)=O
InChI Key InChIKey=SNYRSILPNZIHHZ-FIXZTSJVSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50019481
Affinity DataKi: 0.230nMAssay Description:Compound was evaluated for the inhibition of [3H]-bremazocine binding to Opioid receptor kappa 1 in guinea pig cerebellum membrane homogenates.More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Compound was evaluated for the inhibition of [3H]DAGO([[3H]-D-Ala,MePhe4,Glyol5]enkephalin) binding to mu sites in rat brain homogenates.More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Compound was evaluated for the inhibition of [3H]DSLET([[3H]-D-Ser2,Leu5,Thr6]enkephalin binding to Opioid receptor delta 1 in rat brain homogenates.More data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Compound was evaluated for the agonistic activity against Opioid receptor mu 1 in guinea pig ileum.More data for this Ligand-Target Pair
Affinity DataIC50: 262nMAssay Description:Compound was evaluated for the agonistic activity against Opioid receptor delta 1 in hamster vas deferens.More data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Compound was evaluated for the agonistic activity against Opioid receptor kappa 1 in rabbit vas deferens.More data for this Ligand-Target Pair