BDBM50024254 CHEMBL125021
SMILES CCOC(=O)c1ccc(cc1)-c1nn(Cc2ccccc2)c2ccccc12
InChI Key InChIKey=LPROLPQTWKDPNU-UHFFFAOYSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50024254
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Northwest Agriculture & Forestry University
Curated by ChEMBL
Northwest Agriculture & Forestry University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at PAR1 in PAR-1-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a...More data for this Ligand-Target Pair
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University
Curated by ChEMBL
Northwest Agriculture & Forestry University
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Antagonist activity PAR4 (unknown origin)More data for this Ligand-Target Pair
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Northwest Agriculture & Forestry University
Curated by ChEMBL
Northwest Agriculture & Forestry University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PAR1 (unknown origin)More data for this Ligand-Target Pair
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University
Curated by ChEMBL
Northwest Agriculture & Forestry University
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a...More data for this Ligand-Target Pair