BDBM50028695 CHEMBL3342688
SMILES NC(=N)NCCC[C@H](NC(=O)c1c[nH]c(n1)C(c1ccccc1)c1ccccc1)C(O)=O
InChI Key InChIKey=VQSBEOLLSPCBBL-KRWDZBQOSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50028695
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 6.31nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataEC50: 130nMAssay Description:Agonist activity against C3AR in HMDMs assessed as increase in intracellular calcium release by Fluo-3 AM dye based FLIPR assay relative to 1 uM C3aMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataEC50: 126nMAssay Description:Agonist activity against C3AR in HMDMs assessed as increase in intracellular calcium release by Fluo-3 AM dye based FLIPR assay relative to 1 uM C3aMore data for this Ligand-Target Pair