BDBM50033112 6-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propylamino}-1,3,5-trimethyl-1H-pyrimidine-2,4-dione::CHEMBL420060::Urapidil-5-methyl

SMILES: COc1ccccc1N1CCN(CCCNc2c(C)c(=O)n(C)c(=O)n2C)CC1

InChI Key: InChIKey=HIHZDNKKIUQQSC-UHFFFAOYSA-N

Data: 24 KI

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 24 hits for monomerid = 50033112   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
5-hydroxytryptamine receptor 1A (Human)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		0.350	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A adrenergic receptor (Bovine)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		0.501	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A adrenergic receptor (Human)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		0.630	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A adrenergic receptor (Rat)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		0.700	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A adrenergic receptor (Guinea pig)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		0.790	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A adrenergic receptor (Guinea pig)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A adrenergic receptor (Human)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		2.30	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A adrenergic receptor (Human)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		4.20	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A adrenergic receptor (Bovine)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		4.40	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A adrenergic receptor (Human)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		10	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1D adrenergic receptor (Human)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		21	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A adrenergic receptor (Guinea pig)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		31.6	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1B adrenergic receptor (Mouse)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		40	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1B adrenergic receptor (Pig)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		63.1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1D adrenergic receptor (Rat)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		96	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1B adrenergic receptor (Pig)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		126	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-2C adrenergic receptor (Human)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		131	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1B adrenergic receptor (Golden hamster)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		180	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1D adrenergic receptor (Rat)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		186	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Alpha-2B adrenergic receptor (Human)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		406	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Alpha-1B adrenergic receptor (Human)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		535	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Alpha-1B adrenergic receptor (Human)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		535	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Alpha-2A adrenergic receptor (Human)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		612	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(2) dopamine receptor (Rat)	BDBM50033112 (Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...) Show SMILES Show InChI	GoogleScholar	UniChem		969	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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