BDBM50043931 CHEMBL3356026

SMILES Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2C#N)cc1

InChI Key InChIKey=LXHSPQDCTKLVDN-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50043931   

TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Sanofi R & D

Curated by ChEMBL
LigandPNGBDBM50043931(CHEMBL3356026)
Affinity DataIC50:  6nMAssay Description:Inhibition of human SGK1 using fluo-5(6)-carboxyfluorescein)-RPRAATF-NH2 fluorescently labeled peptide by substrate phosphorylation assay in presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Sanofi R & D

Curated by ChEMBL
LigandPNGBDBM50043931(CHEMBL3356026)
Affinity DataIC50:  199nMAssay Description:Inhibition of human SGK1 using fluo-5(6)-carboxyfluorescein)-RPRAATF-NH2 fluorescently labeled peptide by substrate phosphorylation assay in presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed