BDBM50054761 CHEMBL143767::Trifluoro-methanesulfonic acid 3-(2-dimethylamino-ethyl)-1H-indol-5-yl ester
SMILES CN(C)CCc1c[nH]c2ccc(OS(=O)(=O)C(F)(F)F)cc12
InChI Key InChIKey=HWRKZNBGZMBBTP-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50054761
Affinity DataKi: 3.20nMAssay Description:Compound was tested for binding affinity against cloned human 5-hydroxytryptamine 1D receptor alpha expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Compound was tested for intrinsic efficacy against human 5-hydroxytryptamine 1D receptor beta measured as the reduction of forskolin-stimulated cAMP.More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Compound was tested for intrinsic efficacy against human 5-hydroxytryptamine 1D receptor alpha measured as the reduction of forskolin-stimulated cAMP...More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Compound was tested for binding affinity against cloned human 5-hydroxytryptamine 1D receptor beta expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Compound was tested for binding affinity against cloned human 5-hydroxytryptamine 1A receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataKi: 538nMAssay Description:Compound was tested for binding affinity against cloned human dopamine D2 receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 8.40nMAssay Description:Compound was tested for binding affinity against human 5-hydroxytryptamine 1D receptor alpha clones expressed in human embryonic kidney (HEK 293) cel...More data for this Ligand-Target Pair
Affinity DataIC50: 98nMAssay Description:Compound was tested for binding affinity against human 5-hydroxytryptamine 1D receptor beta clones expressed in human embryonic kidney (HEK 293) cell...More data for this Ligand-Target Pair