BDBM50077028 CHEMBL3416692
SMILES CCCC[C@H](N)C(=O)Nc1cc(ccc1N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)OCc1ccccc1
InChI Key InChIKey=HNWIOZGMMTUVKP-LSYYVWMOSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50077028
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot
Curated by ChEMBL
National Center For Scientific Research&Quot;Demokritos&Quot
Curated by ChEMBL
Affinity DataIC50: 105nMAssay Description:Inhibition of human recombinant IRAP expressed in baculovirus infected cabbage looper ovary Hi5 cells using L-leucine-7-amido-4-methyl coumarin as su...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot
Curated by ChEMBL
National Center For Scientific Research&Quot;Demokritos&Quot
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human recombinant ERAP2 expressed in baculovirus infected cabbage looper ovary Hi5 cells using L-arginyl-7-amido-4-methyl coumarin as s...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Center For Scientific Research&Quot;Demokritos&Quot
Curated by ChEMBL
National Center For Scientific Research&Quot;Demokritos&Quot
Curated by ChEMBL
Affinity DataIC50: 920nMAssay Description:Inhibition of human recombinant ERAP1 expressed in baculovirus infected Sf9 cells using L-leucine-7-amido-4-methyl coumarin as substrate after 5 to 1...More data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Mus musculus)
National Center For Scientific Research&Quot;Demokritos&Quot
Curated by ChEMBL
National Center For Scientific Research&Quot;Demokritos&Quot
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of mouse recombinant IRAP using L-leucine-7-amido-4-methyl coumarin as substrate after 5 to 10 mins by fluorescence assayMore data for this Ligand-Target Pair