BDBM50077112 CHEMBL27812::Cis-(3aR,11bS)-10-Trifluoromethyl-1,2,3,3a,4,5,7,11b-octahydro-5,7-diaza-cyclopenta[a]anthracen-8-one
SMILES FC(F)(F)c1cc(=O)[nH]c2cc3NC[C@@H]4CCC[C@@H]4c3cc12
InChI Key InChIKey=FDZWPAWLXGOXJZ-IUCAKERBSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50077112
Affinity DataKi: 8nMAssay Description:Agonist activity to the human androgen receptor (hAR) in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 9nMAssay Description:Binding affinity to the human androgen receptor (hAR), using [3H]DHT as radioligand in a competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonistic activity against human androgen receptor (hAR) in CV-1 cells using cotransfection assayMore data for this Ligand-Target Pair