BDBM50078630 CHEMBL4296718

SMILES Cn1cc(CCn2cnc(-c3cnn(C)c3)c2-c2ccc(cc2)C#N)cn1

InChI Key InChIKey=RRZVGDGTWNQAPW-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50078630   

TargetBromodomain adjacent to zinc finger domain protein 2A(Human)
Cancer Research Uk Cancer Therapeutics Unit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078630BDBM50078630(CHEMBL4296718)
Affinity DataIC50: 136nMAssay Description:Inhibition of BAZ2A (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
Cancer Research Uk Cancer Therapeutics Unit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078630BDBM50078630(CHEMBL4296718)
Affinity DataIC50: 174nMAssay Description:Displacement of H3K14Ac from BAZ2B (unknown origin) preincubated for 30 mins with non-biotinylated peptide followed by addition of biotinylated pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed