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BDBM50078827 2-(pyridin-3-yl)-1H-benzo[d]imidazole::2-Pyridin-3-yl-1H-benzoimidazole::CHEMBL83103::LDHA Inhibitor, 10

SMILES: c1ccc2[nH]c(nc2c1)-c1cccnc1

InChI Key: InChIKey=BOUOQESVDURNSB-UHFFFAOYSA-N

Data: 4 IC50 2 Kd

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50078827
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
L-lactate dehydrogenase A chain (Rat)	BDBM50078827 (CHEMBL83103 \| LDHA Inhibitor, 10 \| 2-Pyridin-3-yl-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	1.40E+6	n/a	n/a	n/a	7.5	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
L-lactate dehydrogenase A chain (Rat)	BDBM50078827 (CHEMBL83103 \| LDHA Inhibitor, 10 \| 2-Pyridin-3-yl-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>5.00E+5	n/a	n/a	n/a	n/a	7.5	21
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase mTOR (Human)	BDBM50078827 (CHEMBL83103 \| LDHA Inhibitor, 10 \| 2-Pyridin-3-yl-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	4.10E+5	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Methionine aminopeptidase (Escherichia coli (strain K12))	BDBM50078827 (CHEMBL83103 \| LDHA Inhibitor, 10 \| 2-Pyridin-3-yl-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Cytochrome P450 2B1 (Rat)	BDBM50078827 (CHEMBL83103 \| LDHA Inhibitor, 10 \| 2-Pyridin-3-yl-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	2.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Bifunctional epoxide hydrolase 2 (Human)	BDBM50078827 (CHEMBL83103 \| LDHA Inhibitor, 10 \| 2-Pyridin-3-yl-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	9.10E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair