BDBM50088507 CHEBI:63804::CHEMBL1908021

SMILES Oc1ccc(cc1)C1(NC(=O)NC1=O)c1ccccc1

InChI Key InChIKey=XEEDURHPFVXALT-UHFFFAOYSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50088507   

TargetUDP-glucuronosyltransferase 1A1(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50088507(CHEBI:63804 | CHEMBL1908021)
Affinity DataIC50:  1.10E+5nMAssay Description:Inhibition of human recombinant UGT1A1 expressed in HEK293 cells assessed as reduction in estradiol 3-glucuronidation by LC-MS/MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-glucuronosyltransferase 1A1(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50088507(CHEBI:63804 | CHEMBL1908021)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibition of human recombinant UGT1A1 expressed in HEK293 cells assessed as reduction in bilirubin glucuronidation by LC-MS/MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50088507(CHEBI:63804 | CHEMBL1908021)
Affinity DataIC50:  6.42E+4nMAssay Description:Inhibition of human Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50088507(CHEBI:63804 | CHEMBL1908021)
Affinity DataIC50:  4.79E+4nMAssay Description:Inhibition of protein kinase C epsilon expressed in Sf-9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50088507(CHEBI:63804 | CHEMBL1908021)
Affinity DataIC50:  4.06E+4nMAssay Description:Inhibition of human Protein kinase C beta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50088507(CHEBI:63804 | CHEMBL1908021)
Affinity DataIC50:  4.06E+4nMAssay Description:Inhibition of protein kinase C epsilon expressed in Sf-9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed