BDBM50091910 1-Benzyl-4-(2-phenyl-thiazol-4-ylmethyl)-piperazine::CHEMBL64043

SMILES C(N1CCN(Cc2ccccc2)CC1)c1csc(n1)-c1ccccc1

InChI Key InChIKey=SUBIJFYEXXITCD-UHFFFAOYSA-N

Data  5 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50091910   

TargetD(4) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50091910(1-Benzyl-4-(2-phenyl-thiazol-4-ylmethyl)-piperazin...)
Affinity DataKi:  590nMAssay Description:In vitro displacement of [3H]spiperone from the recombinant human dopamine receptor D4 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50091910(1-Benzyl-4-(2-phenyl-thiazol-4-ylmethyl)-piperazin...)
Affinity DataKi:  5.25E+3nMAssay Description:In vitro displacement of [3H]spiperone from the cloned human dopamine receptor D3 stably expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Bovine)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50091910(1-Benzyl-4-(2-phenyl-thiazol-4-ylmethyl)-piperazin...)
Affinity DataKi:  9.20E+3nMAssay Description:In vitro displacement of [3H]- SCH 23390 from the dopamine receptor D1 of bovine striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50091910(1-Benzyl-4-(2-phenyl-thiazol-4-ylmethyl)-piperazin...)
Affinity DataKi:  1.95E+4nMAssay Description:In vitro displacement of [3H]spiperone from the recombinant human dopamine receptor D2L stably expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50091910(1-Benzyl-4-(2-phenyl-thiazol-4-ylmethyl)-piperazin...)
Affinity DataKi:  2.80E+4nMAssay Description:In vitro displacement of [3H]spiperone from the recombinant human dopamine receptor D2L stably expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed