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BDBM50102286 10-benzyl-3-furan-2-yl-10H-benzo[4,5]imidazo[2,1-c][1,2,4]triazin-4-one::CHEMBL113518

SMILES: O=c1c(nnc2n(Cc3ccccc3)c3ccccc3n12)-c1ccco1

InChI Key: InChIKey=LAKWSLSTUWRCOM-UHFFFAOYSA-N

Data: 5 KI 1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50102286
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Adenosine receptor A2b (Human)	BDBM50102286 (10-benzyl-3-furan-2-yl-10H-benzo[4,5]imidazo[2,1-c...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	10	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Adenosine receptor A2a (Human)	BDBM50102286 (10-benzyl-3-furan-2-yl-10H-benzo[4,5]imidazo[2,1-c...) Show SMILES Show InChI	GoogleScholar	UniChem		156	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Adenosine receptor A1 (Bovine)	BDBM50102286 (10-benzyl-3-furan-2-yl-10H-benzo[4,5]imidazo[2,1-c...) Show SMILES Show InChI	GoogleScholar	UniChem		990	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Adenosine receptor A2a (Human)	BDBM50102286 (10-benzyl-3-furan-2-yl-10H-benzo[4,5]imidazo[2,1-c...) Show SMILES Show InChI	GoogleScholar	UniChem		1.24E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Adenosine receptor A3 (Human)	BDBM50102286 (10-benzyl-3-furan-2-yl-10H-benzo[4,5]imidazo[2,1-c...) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Adenosine receptor A1 (Human)	BDBM50102286 (10-benzyl-3-furan-2-yl-10H-benzo[4,5]imidazo[2,1-c...) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair