BDBM50105912 CHEMBL3133762
SMILES Nc1nccc(n1)-c1cn(C(=O)N2CCOCC2)c2ccc(Br)cc12
InChI Key InChIKey=PTQHCVXFSMUUIH-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50105912
TargetDual specificity tyrosine-phosphorylation-regulated kinase 3(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of Dyrk3 (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of Dyrk2 (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair