BDBM50109461 1-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-phenylurea::1-(2-Furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-phenyl-urea::CHEMBL324735::MRE 3046F20
SMILES Cn1cc2c(n1)nc(NC(=O)Nc1ccccc1)n1nc(nc21)-c1ccco1
InChI Key InChIKey=OPNAVJJOJBREBM-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 34 hits for monomerid = 50109461
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]-MRE3008F20 from human recombinant adenosine A3 receptor expressed in HEK293 cells after 120 mins by scintillation counting analy...More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]MRE3008-F20 from human A3 receptor expressed in CHO cells by scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]MRE 3008F20 from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]-MRE3008-F20 from human A3 receptors expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]-MRE3008-F20 from human Adenosine A3 receptor expressed in HEK cells; range 0.13-0.20More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Binding affinity for human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]-MRE 3008-F20 from Human Adenosine A3 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 222nMAssay Description:Displacement of [3H]-DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 222nMAssay Description:Displacement of [3H]-DPCPX from human Adenosine A2B receptor expressed in HEK-293 cells; range 181-273More data for this Ligand-Target Pair
Affinity DataKi: 222nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
Affinity DataKi: 222nMAssay Description:Displacement of [3H]-DPCPX from Human Adenosine A2B receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 222nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A2B receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 222nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cells by scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 381nMAssay Description:Displacement of [3H]-SCH58261 from human recombinant adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation counting analysi...More data for this Ligand-Target Pair
Affinity DataKi: 381nMAssay Description:Displacement of [3H]-ZM-241,385 from human adenosine A2A receptors expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 381nMAssay Description:Displacement of [3H]-ZM 241385 from Human Adenosine A2a receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 381nMAssay Description:Displacement of [3H]-SCH-58,261 from human Adenosine A2A receptor expressed in HEK-293 cells; range 351-415More data for this Ligand-Target Pair
Affinity DataKi: 381nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 381nMAssay Description:Displacement of [3H]ZM-241385 from human A2A receptor expressed in CHO cells by scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 381nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 594nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cells by scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 594nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cell membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 594nMAssay Description:Displacement of [3H]-DPCPX from human Adenosine A1 receptor expressed in CHO cells; range 436-810More data for this Ligand-Target Pair
Affinity DataKi: 594nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 594nMAssay Description:Displacement of [3H]-DPCPX from Human Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 594nMAssay Description:Displacement of [3H]-DPCPX from human Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibitory activity against Human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of IB-MECA agonist-mediated cAMP production in membranes of CHO cells expressing human Adenosine A3 receptorMore data for this Ligand-Target Pair