BDBM50118762 2-(Oxalyl-amino)-4,5,6,7-tetrahydro-benzo[b]thiophene-3-carboxylic acid::2-(carboxyformamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylic acid::2-oxalylamino-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylic acid::CHEMBL138152
SMILES OC(=O)C(=O)Nc1sc2CCCCc2c1C(O)=O
InChI Key InChIKey=ISZAWTJNJSOJQB-UHFFFAOYSA-N
Data 14 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 14 hits for monomerid = 50118762
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Amherst College
Curated by ChEMBL
Amherst College
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of PTP1B I219A mutantMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: 8.10E+3nMAssay Description:Inhibition of PTPN2More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Amherst College
Curated by ChEMBL
Amherst College
Curated by ChEMBL
Affinity DataKi: 8.10E+3nMAssay Description:Binding affinity to PTP1BMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Amherst College
Curated by ChEMBL
Amherst College
Curated by ChEMBL
Affinity DataKi: 8.10E+3nMpH: 5.5Assay Description:Inhibitory effect against recombinant human protein-tyrosine phosphatase 1B (PTP1B), using p-nitrophenyl phosphate substrate at pH 5.5.More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Amherst College
Curated by ChEMBL
Amherst College
Curated by ChEMBL
Affinity DataKi: 8.13E+3nMAssay Description:Binding affinity to human recombinant PTP1BMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase beta(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: 1.90E+4nMAssay Description:Inhibition of PTPRBMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Amherst College
Curated by ChEMBL
Amherst College
Curated by ChEMBL
Affinity DataKi: 3.40E+4nMAssay Description:Inhibition of wild type PTP1BMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase C(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: 4.10E+4nMAssay Description:Inhibition of PTPRCMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase epsilon(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: 4.50E+4nMAssay Description:Inhibition of PTPREMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 6(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: 1.00E+5nMAssay Description:Inhibition of PTPN6More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase alpha(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: 2.90E+5nMAssay Description:Inhibition of PTPRAMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase alpha(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: 2.90E+5nMpH: 5.5Assay Description:Inhibitory effect against human protein-tyrosine phosphatase alpha (PTPalpha), using p-nitrophenyl phosphate substrate at pH 5.5.More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: 4.10E+5nMAssay Description:Inhibition of PTPRFMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: 4.10E+5nMpH: 5.5Assay Description:Inhibitory effect against protein-tyrosine phosphatase Lar, using p-nitrophenyl phosphate as substrate at pH 5.5.More data for this Ligand-Target Pair