BDBM50124610 C-(5-Allyl-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysen-10-yl)-methylamine::CHEMBL8340

SMILES CC1=CC(C)(C)Nc2ccc-3c(C(CC=C)Oc4cccc(CN)c-34)c12

InChI Key InChIKey=NBXZWVNWURAUNV-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50124610   

TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50124610(C-(5-Allyl-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-...)
Affinity DataKi:  140nMAssay Description:Transcriptional repression in HepG2 cells expressing human glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50124610(C-(5-Allyl-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-...)
Affinity DataEC50:  467nMAssay Description:Transcriptional repression in HepG2 cells expressing human glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed