BDBM50128023 CHEMBL3628281

SMILES CC1(C)C2C1C(=O)N(C2=O)c1ccc(NC(=O)c2ccccn2)cc1Cl

InChI Key InChIKey=CEQFGBDWPIJQAJ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50128023   

TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50128023(CHEMBL3628281)
Affinity DataIC50:  140nMAssay Description:Negative allosteric modulation of human mGlu1 receptor in HEK293 cells assessed as potentiation of glutamate-induced calcium mobiliztion by Fluo-4AM ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed