BDBM50128282 3-(1H-Indol-3-yl)-4-[1-(1-methyl-piperidin-4-yl)-1H-indol-3-yl]-pyrrole-2,5-dione::CHEMBL52654

SMILES: CN1CCC(CC1)n1cc(C2=C(C(=O)NC2=O)c2c[nH]c3ccccc23)c2ccccc12

InChI Key: InChIKey=HCJOTKSJPHFVJC-UHFFFAOYSA-N

Data: 11 IC50

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Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 11 hits for monomerid = 50128282   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Protein kinase C eta type (Human)	BDBM50128282 (3-(1H-Indol-3-yl)-4-[1-(1-methyl-piperidin-4-yl)-1...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	40	n/a	n/a	n/a	n/a	n/a	n/a
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Protein kinase C alpha type (Human)	BDBM50128282 (3-(1H-Indol-3-yl)-4-[1-(1-methyl-piperidin-4-yl)-1...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	200	n/a	n/a	n/a	n/a	n/a	n/a
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Protein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type (Rat)	BDBM50128282 (3-(1H-Indol-3-yl)-4-[1-(1-methyl-piperidin-4-yl)-1...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	200	n/a	n/a	n/a	n/a	n/a	n/a
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Protein kinase C beta type (Human)	BDBM50128282 (3-(1H-Indol-3-yl)-4-[1-(1-methyl-piperidin-4-yl)-1...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	20	n/a	n/a	n/a	n/a	n/a	n/a
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Protein kinase C beta type (Human)	BDBM50128282 (3-(1H-Indol-3-yl)-4-[1-(1-methyl-piperidin-4-yl)-1...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	10	n/a	n/a	n/a	n/a	n/a	n/a
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Proto-oncogene tyrosine-protein kinase Src (Human)	BDBM50128282 (3-(1H-Indol-3-yl)-4-[1-(1-methyl-piperidin-4-yl)-1...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	8.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Calcium/calmodulin-dependent protein kinase type II subunit alpha/beta/delta/gamma (Human)	BDBM50128282 (3-(1H-Indol-3-yl)-4-[1-(1-methyl-piperidin-4-yl)-1...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Protein kinase C zeta type (Human)	BDBM50128282 (3-(1H-Indol-3-yl)-4-[1-(1-methyl-piperidin-4-yl)-1...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	5.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Protein kinase C epsilon type (Human)	BDBM50128282 (3-(1H-Indol-3-yl)-4-[1-(1-methyl-piperidin-4-yl)-1...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	50	n/a	n/a	n/a	n/a	n/a	n/a
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Protein kinase C delta type (Human)	BDBM50128282 (3-(1H-Indol-3-yl)-4-[1-(1-methyl-piperidin-4-yl)-1...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	400	n/a	n/a	n/a	n/a	n/a	n/a
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Protein kinase C gamma type (Human)	BDBM50128282 (3-(1H-Indol-3-yl)-4-[1-(1-methyl-piperidin-4-yl)-1...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	500	n/a	n/a	n/a	n/a	n/a	n/a
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