BDBM50128286 3-[1-(1-Isopropyl-piperidin-4-yl)-1H-indol-3-yl]-4-(1-methyl-1H-indol-3-yl)-pyrrole-2,5-dione::CHEMBL301860

SMILES: CC(C)N1CCC(CC1)n1cc(C2=C(C(=O)NC2=O)c2cn(C)c3ccccc23)c2ccccc12

InChI Key: InChIKey=KQUBTSBQLPIFSM-UHFFFAOYSA-N

Data: 10 IC50

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 10 hits for monomerid = 50128286   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Protein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type (Rat)	BDBM50128286 (3-[1-(1-Isopropyl-piperidin-4-yl)-1H-indol-3-yl]-4...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	250	n/a	n/a	n/a	n/a	n/a	n/a
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Protein kinase C alpha type (Human)	BDBM50128286 (3-[1-(1-Isopropyl-piperidin-4-yl)-1H-indol-3-yl]-4...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	340	n/a	n/a	n/a	n/a	n/a	n/a
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Protein kinase C eta type (Human)	BDBM50128286 (3-[1-(1-Isopropyl-piperidin-4-yl)-1H-indol-3-yl]-4...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	130	n/a	n/a	n/a	n/a	n/a	n/a
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Protein kinase C beta type (Human)	BDBM50128286 (3-[1-(1-Isopropyl-piperidin-4-yl)-1H-indol-3-yl]-4...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	26	n/a	n/a	n/a	n/a	n/a	n/a
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Calcium/calmodulin-dependent protein kinase type II subunit alpha/beta/delta/gamma (Human)	BDBM50128286 (3-[1-(1-Isopropyl-piperidin-4-yl)-1H-indol-3-yl]-4...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	7.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Protein kinase C epsilon type (Human)	BDBM50128286 (3-[1-(1-Isopropyl-piperidin-4-yl)-1H-indol-3-yl]-4...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	390	n/a	n/a	n/a	n/a	n/a	n/a
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Protein kinase C delta type (Human)	BDBM50128286 (3-[1-(1-Isopropyl-piperidin-4-yl)-1H-indol-3-yl]-4...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	970	n/a	n/a	n/a	n/a	n/a	n/a
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Protein kinase C beta type (Human)	BDBM50128286 (3-[1-(1-Isopropyl-piperidin-4-yl)-1H-indol-3-yl]-4...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	19	n/a	n/a	n/a	n/a	n/a	n/a
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Protein kinase C gamma type (Human)	BDBM50128286 (3-[1-(1-Isopropyl-piperidin-4-yl)-1H-indol-3-yl]-4...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.30E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Protein kinase C zeta type (Human)	BDBM50128286 (3-[1-(1-Isopropyl-piperidin-4-yl)-1H-indol-3-yl]-4...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	9.30E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair