BDBM50131440 10-(2-(1-methylpiperidin-2-yl)ethyl)-2-(methylsulfinyl)-10H-phenothiazine::2-Methanesulfinyl-10-[2-(1-methyl-piperidin-2-yl)-ethyl]-10H-phenothiazine::CHEMBL1088::MESORIDAZINE::NC-123::Serentil::TPS-23

SMILES: CN1CCCCC1CCN1c2ccccc2Sc2ccc(cc12)S(C)=O

InChI Key: InChIKey=SLVMESMUVMCQIY-UHFFFAOYSA-N

Data: 32 KI  5 IC50

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 37 hits for monomerid = 50131440   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Potassium voltage-gated channel subfamily H member 2 (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	316	n/a	n/a	n/a	n/a	n/a	n/a
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Potassium voltage-gated channel subfamily H member 2 (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	324	n/a	n/a	n/a	n/a	n/a	n/a
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Potassium voltage-gated channel subfamily H member 2 (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	n/a
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Potassium voltage-gated channel subfamily H member 2 (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	320	n/a	n/a	n/a	n/a	n/a	n/a
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Potassium voltage-gated channel subfamily H member 2 (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	324	n/a	n/a	n/a	n/a	n/a	n/a
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Histamine H1 receptor (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		1.80	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Histamine H1 receptor (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		1.81	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A adrenergic receptor (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		2	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A adrenergic receptor (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		2	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(3) dopamine receptor (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		2.60	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(2) dopamine receptor (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		4.30	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 2C (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		4.76	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(2) dopamine receptor (Rat)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 2A (Rat)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		6.30	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 2A (Rat)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		6.30	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 2A (Rat)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		6.30	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(2) dopamine receptor (Rat)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		7.94	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(4) dopamine receptor (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		9.10	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1 (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		10	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(4) dopamine receptor (Rat)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		13.4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M2 (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		15	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(2) dopamine receptor (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		18.9	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(2) dopamine receptor (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		19	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M4 (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		19	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M5 (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		60	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M2 (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		69	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M2 (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		71.4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 7 (Rat)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		73	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 2C (Rat)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		79	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 2C (Rat)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		79.4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M3 (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		90	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 2C (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		157	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 6 (Rat)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		159	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 6 (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		380	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 1A/1B/1D/2C (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		500	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-2A adrenergic receptor (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		1.60E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-2A adrenergic receptor (Human)	BDBM50131440 (CHEMBL1088 | 10-(2-(1-methylpiperidin-2-yl)ethyl)-...) Show SMILES Show InChI	GoogleScholar	UniChem		1.61E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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