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BDBM50132989 4-[3-(6-Methyl-pyridin-2-yl)-1H-pyrazol-4-yl]-quinoline::CHEMBL129677

SMILES: Cc1cccc(n1)-c1n[nH]cc1-c1ccnc2ccccc12

InChI Key: InChIKey=KJTYZDORHCDZPS-UHFFFAOYSA-N

Data: 6 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50132989
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
TGF-beta receptor type-1 (Human)	BDBM50132989 (4-[3-(6-Methyl-pyridin-2-yl)-1H-pyrazol-4-yl]-quin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	34	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
TGF-beta receptor type-1 (Human)	BDBM50132989 (4-[3-(6-Methyl-pyridin-2-yl)-1H-pyrazol-4-yl]-quin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	2.90	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
TGF-beta receptor type-1 (Human)	BDBM50132989 (4-[3-(6-Methyl-pyridin-2-yl)-1H-pyrazol-4-yl]-quin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	7.10	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
TGF-beta receptor type-1 (Human)	BDBM50132989 (4-[3-(6-Methyl-pyridin-2-yl)-1H-pyrazol-4-yl]-quin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	78	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
TGF-beta receptor type-1 (Human)	BDBM50132989 (4-[3-(6-Methyl-pyridin-2-yl)-1H-pyrazol-4-yl]-quin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	25	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
TGF-beta receptor type-1 (Human)	BDBM50132989 (4-[3-(6-Methyl-pyridin-2-yl)-1H-pyrazol-4-yl]-quin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	25	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair