BDBM50147085 7-METHOXY-8-[1-(METHYLSULFONYL)-1H-PYRAZOL-4-YL]NAPHTHALENE-2-CARBOXIMIDAMIDE::7-methoxy-8-(1-(methylsulfonyl)-1H-pyrazol-4-yl)-2-naphthimidamide::8-(1-Methanesulfonyl-1H-pyrazol-4-yl)-7-methoxy-naphthalene-2-carboxamidine::CHEMBL321944::uPa_13

SMILES: COc1ccc2ccc(cc2c1-c1cnn(c1)S(C)(=O)=O)C(N)=N

InChI Key: InChIKey=KQUXAFOLFXHVQN-UHFFFAOYSA-N

Data: 9 KI

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 50147085   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Urokinase-type plasminogen activator (Human)	BDBM50147085 (uPa_13 | 8-(1-Methanesulfonyl-1H-pyrazol-4-yl)-7-m...) Show SMILES Show InChI	GoogleScholar	UniChem		630	-8.45	n/a	n/a	n/a	n/a	n/a	7.4	25
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Urokinase-type plasminogen activator [179-424,C299A,N323Q] (Human)	BDBM50147085 (uPa_13 | 8-(1-Methanesulfonyl-1H-pyrazol-4-yl)-7-m...) Show SMILES Show InChI	GoogleScholar	UniChem		630	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Urokinase-type plasminogen activator (Human)	BDBM50147085 (uPa_13 | 8-(1-Methanesulfonyl-1H-pyrazol-4-yl)-7-m...) Show SMILES Show InChI	GoogleScholar	UniChem		630	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Urokinase-type plasminogen activator (Human)	BDBM50147085 (uPa_13 | 8-(1-Methanesulfonyl-1H-pyrazol-4-yl)-7-m...) Show SMILES Show InChI	GoogleScholar	UniChem		631	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Serine protease 1 (Human)	BDBM50147085 (uPa_13 | 8-(1-Methanesulfonyl-1H-pyrazol-4-yl)-7-m...) Show SMILES Show InChI	GoogleScholar	UniChem		2.70E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Prothrombin (Human)	BDBM50147085 (uPa_13 | 8-(1-Methanesulfonyl-1H-pyrazol-4-yl)-7-m...) Show SMILES Show InChI	GoogleScholar	UniChem		7.10E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Plasminogen (Human)	BDBM50147085 (uPa_13 | 8-(1-Methanesulfonyl-1H-pyrazol-4-yl)-7-m...) Show SMILES Show InChI	GoogleScholar	UniChem		8.50E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Kallikrein-1 (Human)	BDBM50147085 (uPa_13 | 8-(1-Methanesulfonyl-1H-pyrazol-4-yl)-7-m...) Show SMILES Show InChI	GoogleScholar	UniChem		1.40E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Tissue-type plasminogen activator (Human)	BDBM50147085 (uPa_13 | 8-(1-Methanesulfonyl-1H-pyrazol-4-yl)-7-m...) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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