BDBM50152116 CHEMBL3781131

SMILES C[C@]12CCC(C1)C(C)(C)C2NC(=O)c1nn(c-2c1Cc1cc(ccc-21)C1CC1)-c1ccc(Cl)cc1Cl

InChI Key InChIKey=DXHUAQFMQWIMBW-SVANQLSFSA-N

Data  2 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50152116   

TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50152116(CHEMBL3781131)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293-EBNA cell membrane incubated for 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50152116(CHEMBL3781131)
Affinity DataKi: >4.00E+4nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293-EBNA cell membrane incubated for 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50152116(CHEMBL3781131)
Affinity DataIC50:  80nMAssay Description:Antagonist/inverse agonist activity at human CB2 receptors expressed in human Chem4 cell membrane incubated for 30 mins by [35S]GTPgammaS binding ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed