BDBM50170155 CHEMBL3805220
SMILES N#C\N=C(\NCCSc1ccccc1)NC[C@@H]1CC[C@H](C1)c1c[nH]cn1
InChI Key InChIKey=MMZLYDNVAYWZLR-HZPDHXFCSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50170155
Affinity DataKi: 590nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in sf9 cell membrane co-expressing mammalian Galphai2 and Gbet...More data for this Ligand-Target Pair
Affinity DataKi: 1.05E+3nMAssay Description:Displacement of [3H]UR-PI294 from human histamine H4 receptor expressed in sf9 cell membrane co-expressing mammalian Galphai2 and Gbeta1gamma2 incuba...More data for this Ligand-Target Pair
Affinity DataKi: 7.91E+3nMAssay Description:Displacement of [3H]mepyramine from human histamine H1 receptor expressed in sf9 cell membrane co-expressing RGS4 incubated for 60 mins by liquid sci...More data for this Ligand-Target Pair
Affinity DataKi: 9.82E+3nMAssay Description:Displacement of [3H]tiotidine from human histamine H2 receptor expressed in sf9 cell membrane co-expressing Gsalphas incubated for 60 mins by liquid ...More data for this Ligand-Target Pair
Affinity DataEC50: 500nMAssay Description:Agonist activity at human SF-His6-tagged histamine H4 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated response incu...More data for this Ligand-Target Pair
Affinity DataEC50: 589nMAssay Description:Agonist activity at mouse SF-His6-tagged histamine H4 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated response incu...More data for this Ligand-Target Pair