BDBM50173136 CHEMBL2147142

SMILES Cc1noc(Cn2nc3ccc(cn3c2=O)-c2ccc(Oc3ccc(Cl)cc3)cc2)n1

InChI Key InChIKey=WWFCNKUCFKPXRI-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50173136   

TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50173136(CHEMBL2147142)
Affinity DataIC50:  1.34E+5nMAssay Description:Inhibition of 0.1 Hz stimulated human Nav1.5alpha expressed in HEK293 cells assessed as inhibition of late sodium current with 3 compound additions f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed