BDBM50174858 4-(3-Bromo-8-chloro-6,11-dihydro-5H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-yl)-1-[2-(4-chloro-phenyl)-acetyl]-piperazine-2-carboxylic acid methylamide::CHEMBL200851

SMILES CNC(=O)C1CN(CCN1C(=O)Cc1ccc(Cl)cc1)C1c2ccc(Cl)cc2CCc2cc(Br)cnc12

InChI Key InChIKey=WYSDEQZPJKRKGQ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50174858   

TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50174858(4-(3-Bromo-8-chloro-6,11-dihydro-5H-benzo[5,6]cycl...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against human farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed