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BDBM50175248 CHEMBL200586::methyl 3-methyl-1H-thieno[2,3-c]pyrazole-5-carboxylate

SMILES: COC(=O)c1cc2c(C)n[nH]c2s1

InChI Key: InChIKey=MWEIZALZQKSIDX-UHFFFAOYSA-N

Data: 4 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50175248
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Serine/threonine-protein kinase PAK 4 (Human)	BDBM50175248 (methyl 3-methyl-1H-thieno[2,3-c]pyrazole-5-carboxy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Human)	BDBM50175248 (methyl 3-methyl-1H-thieno[2,3-c]pyrazole-5-carboxy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Human)	BDBM50175248 (methyl 3-methyl-1H-thieno[2,3-c]pyrazole-5-carboxy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	2.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase (Human)	BDBM50175248 (methyl 3-methyl-1H-thieno[2,3-c]pyrazole-5-carboxy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair