BDBM50180925 11-methyl-11-aza-tricyclo[12.4.0.03,8]octadeca-1(18),3(8),4,6,14,16-hexaene::7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine::CHEMBL201525
SMILES CN1CCc2ccccc2Cc2ccccc2CC1
InChI Key InChIKey=BXOLXXSMCLYDNG-UHFFFAOYSA-N
Data 14 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 14 hits for monomerid = 50180925
Affinity DataKi: 3.09nMAssay Description:Inhibition of binding to human D5 receptor expressed in HEK 293 cells by functional calcium assayMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 3.47nMAssay Description:Displacement of [3H]SCH23390 from human cloned dopamine D1 receptorMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Inhibition of binding to human D1 receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H]SCH 23390 from human cloned dopamine D1 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.47nMAssay Description:Inhibition of binding to human D2L receptor expressed in HEK 293 cells by functional calcium assayMore data for this Ligand-Target Pair
Affinity DataKi: 11.2nMAssay Description:Binding affinity to human cloned dopamine D5 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11.2nMAssay Description:Inhibition of binding to human D5 receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 40.4nMAssay Description:Inhibition of binding to human D1 receptor expressed in HEK 293 cells by functional calcium assayMore data for this Ligand-Target Pair
Affinity DataKi: 47.5nMAssay Description:Inhibition of binding to human D3 receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 52.5nMAssay Description:Binding affinity to human cloned dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 56.5nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 56.5nMAssay Description:Inhibition of binding to human D2L receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 58.9nMAssay Description:Displacement of [3H]SCH23390 from human cloned dopamine D2L receptorMore data for this Ligand-Target Pair
Affinity DataKi: 134nMAssay Description:Inhibition of binding to human D4 receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair