BDBM50184806 1-((3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl)-4-phenylpiperazine::CHEMBL208018

SMILES Cc1nn(cc1CN1CCN(CC1)c1ccccc1)-c1ccccc1

InChI Key InChIKey=KMPUUVTZQFSTEA-UHFFFAOYSA-N

Data  5 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50184806   

TargetD(4) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50184806(1-((3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl)-4-ph...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50184806(1-((3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl)-4-ph...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2(short) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50184806(1-((3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl)-4-ph...)
Affinity DataKi:  71nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2(long) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50184806(1-((3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl)-4-ph...)
Affinity DataKi:  360nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Pig)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50184806(1-((3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl)-4-ph...)
Affinity DataKi:  3.90E+3nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1 receptor in porcine striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed