BDBM50185368 CHEMBL2371910::CHEMBL439884::Pim[-Trp-Arg-Nva-Arg-Tyr-NH2]2
SMILES CCC[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](N)CCC[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCC)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccc(O)cc1)C(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccc(O)cc1)C(N)=O
InChI Key InChIKey=LTYROZHCAWVGIV-CTAKNGSMSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50185368
Affinity DataKi: 4.10nMAssay Description:Displacement of [125I]hPP from human NPY4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Reduced farnesylation of H-ras transformed NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Displacement of [125I]NPY from human NPY1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibitory activity against Opioid receptor kappa 1 expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:In vitro inhibitory activity against Factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Displacement of [125I]NPY from human NPY2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Inhibitory activity against Opioid receptor kappa 1 expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Inhibition of [3H]-FPP incorporation into biotin-linked K-ras decapeptide (CVLL) by bovine geranygeranyltransferaseMore data for this Ligand-Target Pair