Search and Browse
Download
Enter Data
BDBM50188732 1-cyclopropyl-1-((5-(6-((4-methylpiperazin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)thiophen-2-yl)methyl)-3-m-tolylurea::CHEMBL214063
SMILES: CN1CCN(Cc2ccc-3c(Cc4c-3n[nH]c4-c3ccc(CN(C4CC4)C(=O)Nc4cccc(C)c4)s3)c2)CC1
InChI Key: InChIKey=SFCSGFUQASTWES-UHFFFAOYSA-N
Data: 4 IC50
| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Mast/stem cell growth factor receptor Kit (Human) | BDBM50188732![]() (1-cyclopropyl-1-((5-(6-((4-methylpiperazin-1-yl)me...) | GoogleScholar | UniChem | n/a | n/a | 136 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Vascular endothelial growth factor receptor 2 (Human) | BDBM50188732![]() (1-cyclopropyl-1-((5-(6-((4-methylpiperazin-1-yl)me...) | GoogleScholar | UniChem | n/a | n/a | 171 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Vascular endothelial growth factor receptor 1 (Human) | BDBM50188732![]() (1-cyclopropyl-1-((5-(6-((4-methylpiperazin-1-yl)me...) | GoogleScholar | UniChem | n/a | n/a | 38 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Vascular endothelial growth factor receptor 2 (Human) | BDBM50188732![]() (1-cyclopropyl-1-((5-(6-((4-methylpiperazin-1-yl)me...) | GoogleScholar | UniChem | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||