BDBM50193882 CHEMBL220912::N1-(7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-yl)-N4,N4-dimethylbenzene-1,4-diamine::US8481536, 375

SMILES CN(C)c1ccc(Nc2nnc3cc(cc(C)c3n2)-c2c(C)cccc2C)cc1

InChI Key InChIKey=BSNNWHSHJOIQJN-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50193882   

TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Targegen

Curated by ChEMBL
LigandPNGBDBM50193882(CHEMBL220912 | N1-(7-(2,6-dimethylphenyl)-5-methyl...)
Affinity DataIC50:  240nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Targegen

Curated by ChEMBL
LigandPNGBDBM50193882(CHEMBL220912 | N1-(7-(2,6-dimethylphenyl)-5-methyl...)
Affinity DataIC50:  244nMT: 2°CAssay Description:Testing of inhibition of kinases in vitro using luciferase-based assay from KinaseGlo, Promega Corp.More data for this Ligand-Target Pair
In DepthDetails US Patent