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BDBM50194237 CHEMBL377960::H-Dmt-Tic-NH-CH[(CH2)4-NH2]-Bid

SMILES: Cc1cc(O)cc(C)c1CC(N)C(=O)N1Cc2ccccc2CC1C(=O)NC(CCCCN)c1nc2ccccc2[nH]1

InChI Key: InChIKey=GDHJQGJCKHJHHZ-UHFFFAOYSA-N

Data: 2 KI 2 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50194237
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Delta-type opioid receptor (Mouse)	BDBM50194237 (H-Dmt-Tic-NH-CH[(CH2)4-NH2]-Bid \| CHEMBL377960) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Mu-type opioid receptor (Guinea pig)	BDBM50194237 (H-Dmt-Tic-NH-CH[(CH2)4-NH2]-Bid \| CHEMBL377960) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	39.7	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Mu-type opioid receptor (Rat)	BDBM50194237 (H-Dmt-Tic-NH-CH[(CH2)4-NH2]-Bid \| CHEMBL377960) Show SMILES Show InChI	GoogleScholar	UniChem		0.160	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Delta-type opioid receptor (Rat)	BDBM50194237 (H-Dmt-Tic-NH-CH[(CH2)4-NH2]-Bid \| CHEMBL377960) Show SMILES Show InChI	GoogleScholar	UniChem		0.490	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair