BDBM50194951 2-methyl-3-(6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyridin-3-yl)propanoic acid::CHEMBL218117

SMILES CC(Cc1ccc(OCCc2nc(oc2C)-c2ccccc2)nc1)C(O)=O

InChI Key InChIKey=XKLUVXAVDPISGS-UHFFFAOYSA-N

Data  1 KI  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50194951   

TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194951(2-methyl-3-(6-(2-(5-methyl-2-phenyloxazol-4-yl)eth...)
Affinity DataKi:  2.10E+3nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194951(2-methyl-3-(6-(2-(5-methyl-2-phenyloxazol-4-yl)eth...)
Affinity DataEC50:  3.00E+3nMAssay Description:Displacement of radiolabeled GW2331 from human PPAR alpha by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194951(2-methyl-3-(6-(2-(5-methyl-2-phenyloxazol-4-yl)eth...)
Affinity DataEC50:  287nMAssay Description:Agonist activity at human PPAR alpha in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194951(2-methyl-3-(6-(2-(5-methyl-2-phenyloxazol-4-yl)eth...)
Affinity DataEC50:  268nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed