BDBM50195699 5-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-ethoxy]-8-(2-carboxy-ethyl)-3,4-dihydro-1H-isoquinoline-2-carboxylic acid propyl ester::CHEMBL219836

SMILES CCCOC(=O)N1CCc2c(OCCc3nc(oc3C)-c3ccc(cc3)-c3ccccc3)ccc(CCC(O)=O)c2C1

InChI Key InChIKey=LLUZQFNWHGWRKI-UHFFFAOYSA-N

Data  1 IC50  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50195699   

TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50195699(5-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-ethoxy...)
Affinity DataEC50:  2.75E+3nMAssay Description:Activity at PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50195699(5-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-ethoxy...)
Affinity DataEC50:  2.39E+3nMAssay Description:Displacement of tritium labeled ligand from human PPARalpha by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50195699(5-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-ethoxy...)
Affinity DataEC50:  3nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50195699(5-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-ethoxy...)
Affinity DataIC50:  21nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed