BDBM50205828 CHEMBL220219::CHEMBL373796::H-Tyr-c[D-Allylgly-Gly-Phe-D-Allylgly]NH2

SMILES N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H]1CC=CC[C@@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)CNC1=O)C(N)=O

InChI Key InChIKey=UYBFKIDGDVZVFM-UHFFFAOYSA-N

Data  6 KI  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 10 hits for monomerid = 50205828   

TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  1.05nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  1.92nMAssay Description:Displacement of [3H]DSLET from rat brain delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  2.27nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataIC50: 4.38nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataIC50: 5.63nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  7.04nMAssay Description:Displacement of [3H]DSLET from rat brain delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataIC50: 9.91nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataIC50: 11.9nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  30.4nMAssay Description:Displacement of [3H]U-69593 from guinea pig brain kappa opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  498nMAssay Description:Displacement of [3H]U-69593 from guinea pig brain kappa opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed