BDBM50224478 (1S,5S)-3-(5,6-dibromopyridin-3-yl)-3,6-diazabicyclo[3.2.0]-heptane::CHEMBL393247

SMILES Brc1cc(cnc1Br)N1C[C@@H]2CN[C@@H]2C1

InChI Key InChIKey=GVVFNYMGPONAFJ-IMTBSYHQSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50224478   

TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Neuroscience Research

Curated by ChEMBL
LigandPNGBDBM50224478((1S,5S)-3-(5,6-dibromopyridin-3-yl)-3,6-diazabicyc...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at recombinant human alpha-4-beta-2 nAChR expressed in HEK293 cells assessed as induction of calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed