BDBM50229425 CHEMBL401142::Tyr-(R)-spiro-Aba-Gly-Phe-NH2
SMILES N[C@@H](Cc1ccc(O)cc1)C(=O)N1CCC[C@]11Cc2ccccc2CN(CC(=O)N[C@@H](Cc2ccccc2)C(N)=O)C1=O
InChI Key InChIKey=XXSVWIUHNDWFND-NTBNWUQQSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50229425
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 0.0293nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain after 45 minsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: >10nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Wistar rat brain after 45 minsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(MOUSE)
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 49.8nMAssay Description:Agonist activity at mu opioid receptor in NMRI mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair