BDBM50231056 5-tert-butyl-2-(4-tert-butylphenyl)-1H-indole::CHEMBL254461

SMILES CC(C)(C)c1ccc(cc1)-c1cc2cc(ccc2[nH]1)C(C)(C)C

InChI Key InChIKey=PBUKGCUQLQWIQX-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50231056   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Pfizer

Curated by ChEMBL

LigandBDBM50231056(5-tert-butyl-2-(4-tert-butylphenyl)-1H-indole | CH...)Copy SMILESCopy InChI

Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced calcium influx in HEK293 cellsMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL