BDBM50231061 CHEMBL398275::N-(2-(1H-indol-3-yl)ethyl)-4-(trifluoromethyl)benzamide

SMILES FC(F)(F)c1ccc(cc1)C(=O)NCCc1c[nH]c2ccccc12

InChI Key InChIKey=DLNMLPGZHDNQEL-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50231061   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Pfizer

Curated by ChEMBL

LigandBDBM50231061(N-(2-(1H-indol-3-yl)ethyl)-4-(trifluoromethyl)benz...)Copy SMILESCopy InChI

Affinity DataIC50: 4.23E+3nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced calcium influx in HEK293 cellsMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
Entry Details Article
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