BDBM50231112 2-(4-tert-butylcyclohexyl)-5-(trifluoromethoxy)-1H-benzo[d]imidazole::CHEMBL442442

SMILES CC(C)(C)C1CCC(CC1)c1nc2ccc(OC(F)(F)F)cc2[nH]1

InChI Key InChIKey=DGGBFXCHUUBZED-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50231112   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Pfizer

Curated by ChEMBL

LigandBDBM50231112(2-(4-tert-butylcyclohexyl)-5-(trifluoromethoxy)-1H...)Copy SMILESCopy InChI

Affinity DataIC50: 4.97E+3nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced calcium influx in HEK293 cellsMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
Entry Details Article
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