BDBM50232478 CHEMBL403233
SMILES O[C@@]12CC\C=C/CCCCN3CC[C@@H](C(=C1)c1nccc4c5ccccc5[nH]c14)[C@]1(C[C@@H]4\C=C/CCCCN4[C@@H]21)C3
InChI Key InChIKey=FUCSLKWLLSEMDQ-MKYGIPPKSA-N
Data 12 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 12 hits for monomerid = 50232478
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of human recombinant GSKbetaMore data for this Ligand-Target Pair
Affinity DataIC50: 4.80E+3nMAssay Description:Non-competitive inhibition of human microsomal ACAT2 overexpressed in CHO cells using [14C]oleoyl-CoA as substrate assessed as formation of cholester...More data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+3nMAssay Description:Non-competitive inhibition of human microsomal ACAT1 overexpressed in CHO cells using [14C]oleoyl-CoA as substrate assessed as formation of cholester...More data for this Ligand-Target Pair
Affinity DataIC50: 6.40E+3nMAssay Description:Non-competitive inhibition of microsomal ACAT in human MDM using [14C]oleoyl-CoA as substrate assessed as formation of cholesteryl [14C]-oleate after...More data for this Ligand-Target Pair
Affinity DataIC50: >1.50E+5nMAssay Description:Inhibition of Staphylococcus aureus ATCC 6538p SortA expressed in Escherichia coli using Dabcyl-QALPETGEE-Edans as substrate after 1 hr by fluorescen...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of GSK3alphaMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 1.02E+4nMAssay Description:Non-ATP competitive inhibition of GSK3betaMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human recombinant CDK5/p35More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of recombinant GSK3-beta by ELISAMore data for this Ligand-Target Pair