BDBM50233222 CHEMBL4082248
SMILES CCCCCCCCCC[C@@H]1NC(=N)N[C@]2(CCCO2)[C@@H]1C(O)=O
InChI Key InChIKey=XQIBJGYYXKVIHB-MPGHIAIKSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50233222
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
Tohoku University
Curated by ChEMBL
Tohoku University
Curated by ChEMBL
Affinity DataIC50: 7.5nMAssay Description:Antagonist activity at human Nav1.2 expressed in HEK293T cells assessed as inhibition of VTD-induced sustained current by whole cell patch clamp meth...More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
Tohoku University
Curated by ChEMBL
Tohoku University
Curated by ChEMBL
Affinity DataEC50: 79nMAssay Description:Inhibition of Nav1.2 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
Tohoku University
Curated by ChEMBL
Tohoku University
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Antagonist activity at human Nav1.2 expressed in HEK293T cells assessed as inhibition of VTD-induced tail current by whole cell patch clamp method re...More data for this Ligand-Target Pair